Protein Targets


ProteinProtein nameOrganismSymbolGeneUniProtChEMBLCompounds
5-hydroxytryptamine receptor 1A Homo sapiens; Human5HT1A_HUMANHTR1AP08908 CHEMBL214 7785 / 8305
5-hydroxytryptamine receptor 1B Homo sapiens; Human5HT1B_HUMANHTR1BP28222 CHEMBL1898 2187 / 2333
5-hydroxytryptamine receptor 1D Homo sapiens; Human5HT1D_HUMANHTR1DP28221 CHEMBL1983 2406 / 2500
5-hydroxytryptamine receptor 1E Homo sapiens; Human5HT1E_HUMANHTR1EP28566 CHEMBL2182 350 / 375
5-hydroxytryptamine receptor 1F Homo sapiens; Human5HT1F_HUMANHTR1FP30939 CHEMBL1805 211 / 221
5-hydroxytryptamine receptor 2A Homo sapiens; Human5HT2A_HUMANHTR2AP28223 CHEMBL224 7198 / 9017
5-hydroxytryptamine receptor 2B Homo sapiens; Human5HT2B_HUMANHTR2BP41595 CHEMBL1833 3498 / 5209
5-hydroxytryptamine receptor 2C Homo sapiens; Human5HT2C_HUMANHTR2CP28335 CHEMBL225 6265 / 8045
5-hydroxytryptamine receptor 4 Homo sapiens; Human5HT4R_HUMANHTR4Q13639 CHEMBL1875 1508 / 1615
5-hydroxytryptamine receptor 5A Homo sapiens; Human5HT5A_HUMANHTR5AP47898 CHEMBL3426 854 / 909
5-hydroxytryptamine receptor 6 Homo sapiens; Human5HT6R_HUMANHTR6P50406 CHEMBL3371 6033 / 7813
5-hydroxytryptamine receptor 7 Homo sapiens; Human5HT7R_HUMANHTR7P34969 CHEMBL3155 3310 / 3424
adenosine A1 receptor Homo sapiens; HumanAA1R_HUMANADORA1P30542 CHEMBL226 11337 / 13635
adenosine A2a receptor Homo sapiens; HumanAA2AR_HUMANADORA2AP29274 CHEMBL251 10444 / 12547
adenosine A2b receptor Homo sapiens; HumanAA2BR_HUMANADORA2BP29275 CHEMBL255 5570 / 5928
adenosine A3 receptor Homo sapiens; HumanAA3R_HUMANADORA3P0DMS8 CHEMBL256 9416 / 11579
cholinergic receptor muscarinic 1 Homo sapiens; HumanACM1_HUMANCHRM1P11229 CHEMBL216 6067 / 7941
cholinergic receptor muscarinic 2 Homo sapiens; HumanACM2_HUMANCHRM2P08172 CHEMBL211 4042 / 5888
cholinergic receptor muscarinic 3 Homo sapiens; HumanACM3_HUMANCHRM3P20309 CHEMBL245 3705 / 5460
cholinergic receptor muscarinic 4 Homo sapiens; HumanACM4_HUMANCHRM4P08173 CHEMBL1821 2701 / 4506
cholinergic receptor muscarinic 5 Homo sapiens; HumanACM5_HUMANCHRM5P08912 CHEMBL2035 1999 / 3776
melanocortin 2 receptor Homo sapiens; HumanACTHR_HUMANMC2RQ01718 CHEMBL1965 32 / 34
adrenoceptor alpha 1D Homo sapiens; HumanADA1D_HUMANADRA1DP25100 CHEMBL223 2075 / 3767
adrenoceptor alpha 2A Homo sapiens; HumanADA2A_HUMANADRA2AP08913 CHEMBL1867 1977 / 3616
adrenoceptor alpha 2B Homo sapiens; HumanADA2B_HUMANADRA2BP18089 CHEMBL1942 1170 / 2799
adrenoceptor alpha 2C Homo sapiens; HumanADA2C_HUMANADRA2CP18825 CHEMBL1916 1557 / 3216
adrenoceptor beta 1 Homo sapiens; HumanADRB1_HUMANADRB1P08588 CHEMBL213 2799 / 4676
adrenoceptor beta 2 Homo sapiens; HumanADRB2_HUMANADRB2P07550 CHEMBL210 5497 / 7471
adrenoceptor beta 3 Homo sapiens; HumanADRB3_HUMANADRB3P13945 CHEMBL246 3497 / 5261
angiotensin II receptor type 2 Homo sapiens; HumanAGTR2_HUMANAGTR2P50052 CHEMBL4607 602 / 2371
bradykinin receptor B2 Homo sapiens; HumanBKRB2_HUMANBDKRB2P30411 CHEMBL3157 997 / 2777
calcitonin receptor Homo sapiens; HumanCALCR_HUMANCALCRP30988 CHEMBL1832 61 / 1803
cholecystokinin A receptor Homo sapiens; HumanCCKAR_HUMANCCKARP32238 CHEMBL1901 1217 / 3023
C-C motif chemokine receptor 1 Homo sapiens; HumanCCR1_HUMANCCR1P32246 CHEMBL2413 1355 / 1413
C-C motif chemokine receptor 2 Homo sapiens; HumanCCR2_HUMANCCR2P41597 CHEMBL4015 3296 / 5273
C-C motif chemokine receptor 4 Homo sapiens; HumanCCR4_HUMANCCR4P51679 CHEMBL2414 816 / 2639
C-C motif chemokine receptor 5 (gene/pseudogene) Homo sapiens; HumanCCR5_HUMANCCR5P51681 CHEMBL274 3528 / 5378
cysteinyl leukotriene receptor 1 Homo sapiens; HumanCLTR1_HUMANCYSLTR1Q9Y271 CHEMBL1798 308 / 2043
cannabinoid receptor 1 Homo sapiens; HumanCNR1_HUMANCNR1P21554 CHEMBL218 11737 / 14126
cannabinoid receptor 2 Homo sapiens; HumanCNR2_HUMANCNR2P34972 CHEMBL253 12999 / 13506
C-X-C motif chemokine receptor 1 Homo sapiens; HumanCXCR1_HUMANCXCR1P25024 CHEMBL4029 445 / 2203
C-X-C motif chemokine receptor 2 Homo sapiens; HumanCXCR2_HUMANCXCR2P25025 CHEMBL2434 1484 / 3242
C-X-C motif chemokine receptor 3 Homo sapiens; HumanCXCR3_HUMANCXCR3P49682 CHEMBL4441 1998 / 2117
C-X-C motif chemokine receptor 4 Homo sapiens; HumanCXCR4_HUMANCXCR4P61073 CHEMBL2107 1702 / 1839
dopamine receptor D1 Homo sapiens; HumanDRD1_HUMANDRD1P21728 CHEMBL2056 3441 / 5257
dopamine receptor D2 Homo sapiens; HumanDRD2_HUMANDRD2P14416 CHEMBL217 14743 / 17009
dopamine receptor D3 Homo sapiens; HumanDRD3_HUMANDRD3P35462 CHEMBL234 8248 / 10060
dopamine receptor D4 Homo sapiens; HumanDRD4_HUMANDRD4P21917 CHEMBL219 4262 / 6248
dopamine receptor D5 Homo sapiens; HumanDRD5_HUMANDRD5P21918 CHEMBL1850 735 / 863
endothelin receptor type A Homo sapiens; HumanEDNRA_HUMANEDNRAP25101 CHEMBL252 2187 / 3964
gamma-aminobutyric acid type B receptor subunit 1 Homo sapiens; HumanGABR1_HUMANGABBR1Q9UBS5 CHEMBL2064 30 / 31
cholecystokinin B receptor Homo sapiens; HumanGASR_HUMANCCKBRP32239 CHEMBL298 2410 / 2454
glutamate metabotropic receptor 1 Homo sapiens; HumanGRM1_HUMANGRM1Q13255 CHEMBL3772 2129 / 2202
glutamate metabotropic receptor 2 Homo sapiens; HumanGRM2_HUMANGRM2Q14416 CHEMBL5137 2674 / 2735
glutamate metabotropic receptor 3 Homo sapiens; HumanGRM3_HUMANGRM3Q14832 CHEMBL2888 571 / 614
glutamate metabotropic receptor 4 Homo sapiens; HumanGRM4_HUMANGRM4Q14833 CHEMBL2736 1753 / 1877
glutamate metabotropic receptor 5 Homo sapiens; HumanGRM5_HUMANGRM5P41594 CHEMBL3227 5176 / 5340
glutamate metabotropic receptor 6 Homo sapiens; HumanGRM6_HUMANGRM6O15303 CHEMBL4573 328 / 332
glutamate metabotropic receptor 7 Homo sapiens; HumanGRM7_HUMANGRM7Q14831 CHEMBL3777 232 / 240
glutamate metabotropic receptor 8 Homo sapiens; HumanGRM8_HUMANGRM8O00222 CHEMBL3228 309 / 324
histamine receptor H1 Homo sapiens; HumanHRH1_HUMANHRH1P35367 CHEMBL231 2837 / 4770
histamine receptor H2 Homo sapiens; HumanHRH2_HUMANHRH2P25021 CHEMBL1941 1205 / 2948
histamine receptor H3 Homo sapiens; HumanHRH3_HUMANHRH3Q9Y5N1 CHEMBL264 6414 / 6591
histamine receptor H4 Homo sapiens; HumanHRH4_HUMANHRH4Q9H3N8 CHEMBL3759 3020 / 3169
melanocortin 3 receptor Homo sapiens; HumanMC3R_HUMANMC3RP41968 CHEMBL4644 2240 / 4033
melanocortin 4 receptor Homo sapiens; HumanMC4R_HUMANMC4RP32245 CHEMBL259 6780 / 8611
melanocortin 5 receptor Homo sapiens; HumanMC5R_HUMANMC5RP33032 CHEMBL4608 2286 / 4069
melanocortin 1 receptor Homo sapiens; HumanMSHR_HUMANMC1RQ01726 CHEMBL3795 2267 / 2362
tachykinin receptor 1 Homo sapiens; HumanNK1R_HUMANTACR1P25103 CHEMBL249 4015 / 5821
tachykinin receptor 2 Homo sapiens; HumanNK2R_HUMANTACR2P21452 CHEMBL2327 1484 / 3174
neuropeptides B and W receptor 1 Homo sapiens; HumanNPBW1_HUMANNPBWR1P48145 CHEMBL1293293 541 / 549
neuropeptide FF receptor 1 Homo sapiens; HumanNPFF1_HUMANNPFFR1Q9GZQ6 CHEMBL5951 323 / 336
neuropeptide S receptor 1 Homo sapiens; HumanNPSR1_HUMANNPSR1Q6W5P4 CHEMBL5162 15752 / 15772
neuropeptide Y receptor Y1 Homo sapiens; HumanNPY1R_HUMANNPY1RP25929 CHEMBL4777 1636 / 3470
neuropeptide Y receptor Y2 Homo sapiens; HumanNPY2R_HUMANNPY2RP49146 CHEMBL4018 1183 / 2965
neuropeptide Y receptor Y4 Homo sapiens; HumanNPY4R_HUMANNPY4RP50391 CHEMBL4877 263 / 290
neuropeptide Y receptor Y5 Homo sapiens; HumanNPY5R_HUMANNPY5RQ15761 CHEMBL4561 1511 / 1591
opioid receptor delta 1 Homo sapiens; HumanOPRD_HUMANOPRD1P41143 CHEMBL236 9699 / 11795
opioid receptor kappa 1 Homo sapiens; HumanOPRK_HUMANOPRK1P41145 CHEMBL237 10312 / 12658
opioid receptor mu 1 Homo sapiens; HumanOPRM_HUMANOPRM1P35372 CHEMBL233 10960 / 13295
opioid related nociceptin receptor 1 Homo sapiens; HumanOPRX_HUMANOPRL1P41146 CHEMBL2014 3086 / 3318
platelet activating factor receptor Homo sapiens; HumanPTAFR_HUMANPTAFRP25105 CHEMBL250 796 / 2543
trace amine associated receptor 1 Homo sapiens; HumanTAAR1_HUMANTAAR1Q96RJ0 CHEMBL5857 1327 / 1334
thyroid stimulating hormone receptor Homo sapiens; HumanTSHR_HUMANTSHRP16473 CHEMBL1963 29911 / 29930
arginine vasopressin receptor 1A Homo sapiens; HumanV1AR_HUMANAVPR1AP37288 CHEMBL1889 1723 / 3531
vasoactive intestinal peptide receptor 1 Homo sapiens; HumanVIPR1_HUMANVIPR1P32241 CHEMBL5144 56 / 1800