Protein Targets


ProteinProtein nameOrganismSymbolGeneUniProtChEMBLCompounds
5-hydroxytryptamine receptor 1A Homo sapiens; Human5HT1A_HUMANHTR1AP08908 CHEMBL214 9422 / 10016
5-hydroxytryptamine receptor 1B Homo sapiens; Human5HT1B_HUMANHTR1BP28222 CHEMBL1898 2475 / 2634
5-hydroxytryptamine receptor 1D Homo sapiens; Human5HT1D_HUMANHTR1DP28221 CHEMBL1983 2655 / 2754
5-hydroxytryptamine receptor 1E Homo sapiens; Human5HT1E_HUMANHTR1EP28566 CHEMBL2182 565 / 597
5-hydroxytryptamine receptor 1F Homo sapiens; Human5HT1F_HUMANHTR1FP30939 CHEMBL1805 212 / 222
5-hydroxytryptamine receptor 2A Homo sapiens; Human5HT2A_HUMANHTR2AP28223 CHEMBL224 8589 / 10505
5-hydroxytryptamine receptor 2B Homo sapiens; Human5HT2B_HUMANHTR2BP41595 CHEMBL1833 4230 / 5981
5-hydroxytryptamine receptor 2C Homo sapiens; Human5HT2C_HUMANHTR2CP28335 CHEMBL225 7347 / 9196
5-hydroxytryptamine receptor 4 Homo sapiens; Human5HT4R_HUMANHTR4Q13639 CHEMBL1875 1760 / 1877
5-hydroxytryptamine receptor 5A Homo sapiens; Human5HT5A_HUMANHTR5AP47898 CHEMBL3426 1119 / 1184
5-hydroxytryptamine receptor 6 Homo sapiens; Human5HT6R_HUMANHTR6P50406 CHEMBL3371 6970 / 8783
5-hydroxytryptamine receptor 7 Homo sapiens; Human5HT7R_HUMANHTR7P34969 CHEMBL3155 4455 / 4622
adenosine A1 receptor Homo sapiens; HumanAA1R_HUMANADORA1P30542 CHEMBL226 12364 / 14663
adenosine A2a receptor Homo sapiens; HumanAA2AR_HUMANADORA2AP29274 CHEMBL251 11667 / 13796
adenosine A2b receptor Homo sapiens; HumanAA2BR_HUMANADORA2BP29275 CHEMBL255 6617 / 6983
adenosine A3 receptor Homo sapiens; HumanAA3R_HUMANADORA3P0DMS8 CHEMBL256 10578 / 12770
cholinergic receptor muscarinic 1 Homo sapiens; HumanACM1_HUMANCHRM1P11229 CHEMBL216 6980 / 8900
cholinergic receptor muscarinic 2 Homo sapiens; HumanACM2_HUMANCHRM2P08172 CHEMBL211 4670 / 6568
cholinergic receptor muscarinic 3 Homo sapiens; HumanACM3_HUMANCHRM3P20309 CHEMBL245 4350 / 6109
cholinergic receptor muscarinic 4 Homo sapiens; HumanACM4_HUMANCHRM4P08173 CHEMBL1821 3558 / 5422
cholinergic receptor muscarinic 5 Homo sapiens; HumanACM5_HUMANCHRM5P08912 CHEMBL2035 2416 / 4200
melanocortin 2 receptor Homo sapiens; HumanACTHR_HUMANMC2RQ01718 CHEMBL1965 33 / 35
adrenoceptor alpha 1D Homo sapiens; HumanADA1D_HUMANADRA1DP25100 CHEMBL223 2404 / 4100
adrenoceptor alpha 2A Homo sapiens; HumanADA2A_HUMANADRA2AP08913 CHEMBL1867 2341 / 3984
adrenoceptor alpha 2B Homo sapiens; HumanADA2B_HUMANADRA2BP18089 CHEMBL1942 1450 / 3084
adrenoceptor alpha 2C Homo sapiens; HumanADA2C_HUMANADRA2CP18825 CHEMBL1916 1786 / 3449
adrenoceptor beta 1 Homo sapiens; HumanADRB1_HUMANADRB1P08588 CHEMBL213 3273 / 5152
adrenoceptor beta 2 Homo sapiens; HumanADRB2_HUMANADRB2P07550 CHEMBL210 6371 / 8365
adrenoceptor beta 3 Homo sapiens; HumanADRB3_HUMANADRB3P13945 CHEMBL246 3706 / 5472
angiotensin II receptor type 2 Homo sapiens; HumanAGTR2_HUMANAGTR2P50052 CHEMBL4607 651 / 2421
bradykinin receptor B2 Homo sapiens; HumanBKRB2_HUMANBDKRB2P30411 CHEMBL3157 1048 / 2828
calcitonin receptor Homo sapiens; HumanCALCR_HUMANCALCRP30988 CHEMBL1832 467 / 2215
cholecystokinin A receptor Homo sapiens; HumanCCKAR_HUMANCCKARP32238 CHEMBL1901 1406 / 3226
C-C motif chemokine receptor 1 Homo sapiens; HumanCCR1_HUMANCCR1P32246 CHEMBL2413 1646 / 1704
C-C motif chemokine receptor 2 Homo sapiens; HumanCCR2_HUMANCCR2P41597 CHEMBL4015 3529 / 5515
C-C motif chemokine receptor 4 Homo sapiens; HumanCCR4_HUMANCCR4P51679 CHEMBL2414 980 / 2812
C-C motif chemokine receptor 5 Homo sapiens; HumanCCR5_HUMANCCR5P51681 CHEMBL274 3691 / 5541
cysteinyl leukotriene receptor 1 Homo sapiens; HumanCLTR1_HUMANCYSLTR1Q9Y271 CHEMBL1798 348 / 2083
cannabinoid receptor 1 Homo sapiens; HumanCNR1_HUMANCNR1P21554 CHEMBL218 14060 / 16708
cannabinoid receptor 2 Homo sapiens; HumanCNR2_HUMANCNR2P34972 CHEMBL253 14804 / 15481
C-X-C motif chemokine receptor 1 Homo sapiens; HumanCXCR1_HUMANCXCR1P25024 CHEMBL4029 459 / 2217
C-X-C motif chemokine receptor 2 Homo sapiens; HumanCXCR2_HUMANCXCR2P25025 CHEMBL2434 1521 / 3279
C-X-C motif chemokine receptor 3 Homo sapiens; HumanCXCR3_HUMANCXCR3P49682 CHEMBL4441 2267 / 2386
C-X-C motif chemokine receptor 4 Homo sapiens; HumanCXCR4_HUMANCXCR4P61073 CHEMBL2107 2874 / 3025
dopamine receptor D1 Homo sapiens; HumanDRD1_HUMANDRD1P21728 CHEMBL2056 4538 / 6427
dopamine receptor D2 Homo sapiens; HumanDRD2_HUMANDRD2P14416 CHEMBL217 17907 / 20602
dopamine receptor D3 Homo sapiens; HumanDRD3_HUMANDRD3P35462 CHEMBL234 9435 / 11350
dopamine receptor D4 Homo sapiens; HumanDRD4_HUMANDRD4P21917 CHEMBL219 4850 / 6919
dopamine receptor D5 Homo sapiens; HumanDRD5_HUMANDRD5P21918 CHEMBL1850 1083 / 1223
endothelin receptor type A Homo sapiens; HumanEDNRA_HUMANEDNRAP25101 CHEMBL252 2372 / 4149
gamma-aminobutyric acid type B receptor subunit 1 Homo sapiens; HumanGABR1_HUMANGABBR1Q9UBS5 CHEMBL2064 56 / 57
cholecystokinin B receptor Homo sapiens; HumanGASR_HUMANCCKBRP32239 CHEMBL298 2586 / 2648
glutamate metabotropic receptor 1 Homo sapiens; HumanGRM1_HUMANGRM1Q13255 CHEMBL3772 2162 / 2235
glutamate metabotropic receptor 2 Homo sapiens; HumanGRM2_HUMANGRM2Q14416 CHEMBL5137 2959 / 3023
glutamate metabotropic receptor 3 Homo sapiens; HumanGRM3_HUMANGRM3Q14832 CHEMBL2888 608 / 651
glutamate metabotropic receptor 4 Homo sapiens; HumanGRM4_HUMANGRM4Q14833 CHEMBL2736 2079 / 2208
glutamate metabotropic receptor 5 Homo sapiens; HumanGRM5_HUMANGRM5P41594 CHEMBL3227 5553 / 5718
glutamate metabotropic receptor 6 Homo sapiens; HumanGRM6_HUMANGRM6O15303 CHEMBL4573 343 / 347
glutamate metabotropic receptor 7 Homo sapiens; HumanGRM7_HUMANGRM7Q14831 CHEMBL3777 254 / 262
glutamate metabotropic receptor 8 Homo sapiens; HumanGRM8_HUMANGRM8O00222 CHEMBL3228 322 / 337
histamine receptor H1 Homo sapiens; HumanHRH1_HUMANHRH1P35367 CHEMBL231 3452 / 5410
histamine receptor H2 Homo sapiens; HumanHRH2_HUMANHRH2P25021 CHEMBL1941 1700 / 3476
histamine receptor H3 Homo sapiens; HumanHRH3_HUMANHRH3Q9Y5N1 CHEMBL264 7509 / 7713
histamine receptor H4 Homo sapiens; HumanHRH4_HUMANHRH4Q9H3N8 CHEMBL3759 3548 / 3701
melanocortin 3 receptor Homo sapiens; HumanMC3R_HUMANMC3RP41968 CHEMBL4644 2349 / 4144
melanocortin 4 receptor Homo sapiens; HumanMC4R_HUMANMC4RP32245 CHEMBL259 7103 / 8936
melanocortin 5 receptor Homo sapiens; HumanMC5R_HUMANMC5RP33032 CHEMBL4608 2374 / 4165
melanocortin 1 receptor Homo sapiens; HumanMSHR_HUMANMC1RQ01726 CHEMBL3795 2378 / 2473
tachykinin receptor 1 Homo sapiens; HumanNK1R_HUMANTACR1P25103 CHEMBL249 4191 / 5999
tachykinin receptor 2 Homo sapiens; HumanNK2R_HUMANTACR2P21452 CHEMBL2327 1560 / 3250
neuropeptides B and W receptor 1 Homo sapiens; HumanNPBW1_HUMANNPBWR1P48145 CHEMBL1293293 542 / 550
neuropeptide FF receptor 1 Homo sapiens; HumanNPFF1_HUMANNPFFR1Q9GZQ6 CHEMBL5951 329 / 349
neuropeptide S receptor 1 Homo sapiens; HumanNPSR1_HUMANNPSR1Q6W5P4 CHEMBL5162 15764 / 15784
neuropeptide Y receptor Y1 Homo sapiens; HumanNPY1R_HUMANNPY1RP25929 CHEMBL4777 1894 / 3752
neuropeptide Y receptor Y2 Homo sapiens; HumanNPY2R_HUMANNPY2RP49146 CHEMBL4018 1454 / 3262
neuropeptide Y receptor Y4 Homo sapiens; HumanNPY4R_HUMANNPY4RP50391 CHEMBL4877 772 / 824
neuropeptide Y receptor Y5 Homo sapiens; HumanNPY5R_HUMANNPY5RQ15761 CHEMBL4561 1682 / 1788
opioid receptor delta 1 Homo sapiens; HumanOPRD_HUMANOPRD1P41143 CHEMBL236 10731 / 12871
opioid receptor kappa 1 Homo sapiens; HumanOPRK_HUMANOPRK1P41145 CHEMBL237 11463 / 13975
opioid receptor mu 1 Homo sapiens; HumanOPRM_HUMANOPRM1P35372 CHEMBL233 12998 / 15406
opioid related nociceptin receptor 1 Homo sapiens; HumanOPRX_HUMANOPRL1P41146 CHEMBL2014 3236 / 3473
platelet activating factor receptor Homo sapiens; HumanPTAFR_HUMANPTAFRP25105 CHEMBL250 822 / 2569
trace amine associated receptor 1 Homo sapiens; HumanTAAR1_HUMANTAAR1Q96RJ0 CHEMBL5857 1333 / 1340
thyroid stimulating hormone receptor Homo sapiens; HumanTSHR_HUMANTSHRP16473 CHEMBL1963 29918 / 29937
arginine vasopressin receptor 1A Homo sapiens; HumanV1AR_HUMANAVPR1AP37288 CHEMBL1889 2156 / 3971
vasoactive intestinal peptide receptor 1 Homo sapiens; HumanVIPR1_HUMANVIPR1P32241 CHEMBL5144 148 / 1892