 | 5-hydroxytryptamine receptor 1A | Homo sapiens; Human | 5HT1A_HUMAN | HTR1A | P08908 | CHEMBL214 | 9422 / 10016 |
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 | 5-hydroxytryptamine receptor 1B | Homo sapiens; Human | 5HT1B_HUMAN | HTR1B | P28222 | CHEMBL1898 | 2475 / 2634 |
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 | 5-hydroxytryptamine receptor 1D | Homo sapiens; Human | 5HT1D_HUMAN | HTR1D | P28221 | CHEMBL1983 | 2655 / 2754 |
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 | 5-hydroxytryptamine receptor 1E | Homo sapiens; Human | 5HT1E_HUMAN | HTR1E | P28566 | CHEMBL2182 | 565 / 597 |
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 | 5-hydroxytryptamine receptor 1F | Homo sapiens; Human | 5HT1F_HUMAN | HTR1F | P30939 | CHEMBL1805 | 212 / 222 |
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 | 5-hydroxytryptamine receptor 2A | Homo sapiens; Human | 5HT2A_HUMAN | HTR2A | P28223 | CHEMBL224 | 8589 / 10505 |
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 | 5-hydroxytryptamine receptor 2B | Homo sapiens; Human | 5HT2B_HUMAN | HTR2B | P41595 | CHEMBL1833 | 4230 / 5981 |
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 | 5-hydroxytryptamine receptor 2C | Homo sapiens; Human | 5HT2C_HUMAN | HTR2C | P28335 | CHEMBL225 | 7347 / 9196 |
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 | 5-hydroxytryptamine receptor 4 | Homo sapiens; Human | 5HT4R_HUMAN | HTR4 | Q13639 | CHEMBL1875 | 1760 / 1877 |
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 | 5-hydroxytryptamine receptor 5A | Homo sapiens; Human | 5HT5A_HUMAN | HTR5A | P47898 | CHEMBL3426 | 1119 / 1184 |
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 | 5-hydroxytryptamine receptor 6 | Homo sapiens; Human | 5HT6R_HUMAN | HTR6 | P50406 | CHEMBL3371 | 6970 / 8783 |
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 | 5-hydroxytryptamine receptor 7 | Homo sapiens; Human | 5HT7R_HUMAN | HTR7 | P34969 | CHEMBL3155 | 4455 / 4622 |
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 | adenosine A1 receptor | Homo sapiens; Human | AA1R_HUMAN | ADORA1 | P30542 | CHEMBL226 | 12364 / 14663 |
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 | adenosine A2a receptor | Homo sapiens; Human | AA2AR_HUMAN | ADORA2A | P29274 | CHEMBL251 | 11667 / 13796 |
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 | adenosine A2b receptor | Homo sapiens; Human | AA2BR_HUMAN | ADORA2B | P29275 | CHEMBL255 | 6617 / 6983 |
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 | adenosine A3 receptor | Homo sapiens; Human | AA3R_HUMAN | ADORA3 | P0DMS8 | CHEMBL256 | 10578 / 12770 |
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 | cholinergic receptor muscarinic 1 | Homo sapiens; Human | ACM1_HUMAN | CHRM1 | P11229 | CHEMBL216 | 6980 / 8900 |
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 | cholinergic receptor muscarinic 2 | Homo sapiens; Human | ACM2_HUMAN | CHRM2 | P08172 | CHEMBL211 | 4670 / 6568 |
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 | cholinergic receptor muscarinic 3 | Homo sapiens; Human | ACM3_HUMAN | CHRM3 | P20309 | CHEMBL245 | 4350 / 6109 |
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 | cholinergic receptor muscarinic 4 | Homo sapiens; Human | ACM4_HUMAN | CHRM4 | P08173 | CHEMBL1821 | 3558 / 5422 |
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 | cholinergic receptor muscarinic 5 | Homo sapiens; Human | ACM5_HUMAN | CHRM5 | P08912 | CHEMBL2035 | 2416 / 4200 |
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 | melanocortin 2 receptor | Homo sapiens; Human | ACTHR_HUMAN | MC2R | Q01718 | CHEMBL1965 | 33 / 35 |
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 | adrenoceptor alpha 1D | Homo sapiens; Human | ADA1D_HUMAN | ADRA1D | P25100 | CHEMBL223 | 2404 / 4100 |
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 | adrenoceptor alpha 2A | Homo sapiens; Human | ADA2A_HUMAN | ADRA2A | P08913 | CHEMBL1867 | 2341 / 3984 |
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 | adrenoceptor alpha 2B | Homo sapiens; Human | ADA2B_HUMAN | ADRA2B | P18089 | CHEMBL1942 | 1450 / 3084 |
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 | adrenoceptor alpha 2C | Homo sapiens; Human | ADA2C_HUMAN | ADRA2C | P18825 | CHEMBL1916 | 1786 / 3449 |
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 | adrenoceptor beta 1 | Homo sapiens; Human | ADRB1_HUMAN | ADRB1 | P08588 | CHEMBL213 | 3273 / 5152 |
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 | adrenoceptor beta 2 | Homo sapiens; Human | ADRB2_HUMAN | ADRB2 | P07550 | CHEMBL210 | 6371 / 8365 |
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 | adrenoceptor beta 3 | Homo sapiens; Human | ADRB3_HUMAN | ADRB3 | P13945 | CHEMBL246 | 3706 / 5472 |
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 | angiotensin II receptor type 2 | Homo sapiens; Human | AGTR2_HUMAN | AGTR2 | P50052 | CHEMBL4607 | 651 / 2421 |
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 | bradykinin receptor B2 | Homo sapiens; Human | BKRB2_HUMAN | BDKRB2 | P30411 | CHEMBL3157 | 1048 / 2828 |
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 | calcitonin receptor | Homo sapiens; Human | CALCR_HUMAN | CALCR | P30988 | CHEMBL1832 | 467 / 2215 |
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 | cholecystokinin A receptor | Homo sapiens; Human | CCKAR_HUMAN | CCKAR | P32238 | CHEMBL1901 | 1406 / 3226 |
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 | C-C motif chemokine receptor 1 | Homo sapiens; Human | CCR1_HUMAN | CCR1 | P32246 | CHEMBL2413 | 1646 / 1704 |
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 | C-C motif chemokine receptor 2 | Homo sapiens; Human | CCR2_HUMAN | CCR2 | P41597 | CHEMBL4015 | 3529 / 5515 |
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 | C-C motif chemokine receptor 4 | Homo sapiens; Human | CCR4_HUMAN | CCR4 | P51679 | CHEMBL2414 | 980 / 2812 |
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 | C-C motif chemokine receptor 5 | Homo sapiens; Human | CCR5_HUMAN | CCR5 | P51681 | CHEMBL274 | 3691 / 5541 |
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 | cysteinyl leukotriene receptor 1 | Homo sapiens; Human | CLTR1_HUMAN | CYSLTR1 | Q9Y271 | CHEMBL1798 | 348 / 2083 |
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 | cannabinoid receptor 1 | Homo sapiens; Human | CNR1_HUMAN | CNR1 | P21554 | CHEMBL218 | 14060 / 16708 |
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 | cannabinoid receptor 2 | Homo sapiens; Human | CNR2_HUMAN | CNR2 | P34972 | CHEMBL253 | 14804 / 15481 |
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 | C-X-C motif chemokine receptor 1 | Homo sapiens; Human | CXCR1_HUMAN | CXCR1 | P25024 | CHEMBL4029 | 459 / 2217 |
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 | C-X-C motif chemokine receptor 2 | Homo sapiens; Human | CXCR2_HUMAN | CXCR2 | P25025 | CHEMBL2434 | 1521 / 3279 |
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 | C-X-C motif chemokine receptor 3 | Homo sapiens; Human | CXCR3_HUMAN | CXCR3 | P49682 | CHEMBL4441 | 2267 / 2386 |
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 | C-X-C motif chemokine receptor 4 | Homo sapiens; Human | CXCR4_HUMAN | CXCR4 | P61073 | CHEMBL2107 | 2874 / 3025 |
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 | dopamine receptor D1 | Homo sapiens; Human | DRD1_HUMAN | DRD1 | P21728 | CHEMBL2056 | 4538 / 6427 |
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 | dopamine receptor D2 | Homo sapiens; Human | DRD2_HUMAN | DRD2 | P14416 | CHEMBL217 | 17907 / 20602 |
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 | dopamine receptor D3 | Homo sapiens; Human | DRD3_HUMAN | DRD3 | P35462 | CHEMBL234 | 9435 / 11350 |
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 | dopamine receptor D4 | Homo sapiens; Human | DRD4_HUMAN | DRD4 | P21917 | CHEMBL219 | 4850 / 6919 |
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 | dopamine receptor D5 | Homo sapiens; Human | DRD5_HUMAN | DRD5 | P21918 | CHEMBL1850 | 1083 / 1223 |
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 | endothelin receptor type A | Homo sapiens; Human | EDNRA_HUMAN | EDNRA | P25101 | CHEMBL252 | 2372 / 4149 |
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 | gamma-aminobutyric acid type B receptor subunit 1 | Homo sapiens; Human | GABR1_HUMAN | GABBR1 | Q9UBS5 | CHEMBL2064 | 56 / 57 |
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 | cholecystokinin B receptor | Homo sapiens; Human | GASR_HUMAN | CCKBR | P32239 | CHEMBL298 | 2586 / 2648 |
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 | glutamate metabotropic receptor 1 | Homo sapiens; Human | GRM1_HUMAN | GRM1 | Q13255 | CHEMBL3772 | 2162 / 2235 |
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 | glutamate metabotropic receptor 2 | Homo sapiens; Human | GRM2_HUMAN | GRM2 | Q14416 | CHEMBL5137 | 2959 / 3023 |
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 | glutamate metabotropic receptor 3 | Homo sapiens; Human | GRM3_HUMAN | GRM3 | Q14832 | CHEMBL2888 | 608 / 651 |
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 | glutamate metabotropic receptor 4 | Homo sapiens; Human | GRM4_HUMAN | GRM4 | Q14833 | CHEMBL2736 | 2079 / 2208 |
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 | glutamate metabotropic receptor 5 | Homo sapiens; Human | GRM5_HUMAN | GRM5 | P41594 | CHEMBL3227 | 5553 / 5718 |
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 | glutamate metabotropic receptor 6 | Homo sapiens; Human | GRM6_HUMAN | GRM6 | O15303 | CHEMBL4573 | 343 / 347 |
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 | glutamate metabotropic receptor 7 | Homo sapiens; Human | GRM7_HUMAN | GRM7 | Q14831 | CHEMBL3777 | 254 / 262 |
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 | glutamate metabotropic receptor 8 | Homo sapiens; Human | GRM8_HUMAN | GRM8 | O00222 | CHEMBL3228 | 322 / 337 |
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 | histamine receptor H1 | Homo sapiens; Human | HRH1_HUMAN | HRH1 | P35367 | CHEMBL231 | 3452 / 5410 |
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 | histamine receptor H2 | Homo sapiens; Human | HRH2_HUMAN | HRH2 | P25021 | CHEMBL1941 | 1700 / 3476 |
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 | histamine receptor H3 | Homo sapiens; Human | HRH3_HUMAN | HRH3 | Q9Y5N1 | CHEMBL264 | 7509 / 7713 |
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 | histamine receptor H4 | Homo sapiens; Human | HRH4_HUMAN | HRH4 | Q9H3N8 | CHEMBL3759 | 3548 / 3701 |
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 | melanocortin 3 receptor | Homo sapiens; Human | MC3R_HUMAN | MC3R | P41968 | CHEMBL4644 | 2349 / 4144 |
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 | melanocortin 4 receptor | Homo sapiens; Human | MC4R_HUMAN | MC4R | P32245 | CHEMBL259 | 7103 / 8936 |
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 | melanocortin 5 receptor | Homo sapiens; Human | MC5R_HUMAN | MC5R | P33032 | CHEMBL4608 | 2374 / 4165 |
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 | melanocortin 1 receptor | Homo sapiens; Human | MSHR_HUMAN | MC1R | Q01726 | CHEMBL3795 | 2378 / 2473 |
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 | tachykinin receptor 1 | Homo sapiens; Human | NK1R_HUMAN | TACR1 | P25103 | CHEMBL249 | 4191 / 5999 |
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 | tachykinin receptor 2 | Homo sapiens; Human | NK2R_HUMAN | TACR2 | P21452 | CHEMBL2327 | 1560 / 3250 |
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 | neuropeptides B and W receptor 1 | Homo sapiens; Human | NPBW1_HUMAN | NPBWR1 | P48145 | CHEMBL1293293 | 542 / 550 |
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 | neuropeptide FF receptor 1 | Homo sapiens; Human | NPFF1_HUMAN | NPFFR1 | Q9GZQ6 | CHEMBL5951 | 329 / 349 |
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 | neuropeptide S receptor 1 | Homo sapiens; Human | NPSR1_HUMAN | NPSR1 | Q6W5P4 | CHEMBL5162 | 15764 / 15784 |
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 | neuropeptide Y receptor Y1 | Homo sapiens; Human | NPY1R_HUMAN | NPY1R | P25929 | CHEMBL4777 | 1894 / 3752 |
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 | neuropeptide Y receptor Y2 | Homo sapiens; Human | NPY2R_HUMAN | NPY2R | P49146 | CHEMBL4018 | 1454 / 3262 |
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 | neuropeptide Y receptor Y4 | Homo sapiens; Human | NPY4R_HUMAN | NPY4R | P50391 | CHEMBL4877 | 772 / 824 |
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 | neuropeptide Y receptor Y5 | Homo sapiens; Human | NPY5R_HUMAN | NPY5R | Q15761 | CHEMBL4561 | 1682 / 1788 |
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 | opioid receptor delta 1 | Homo sapiens; Human | OPRD_HUMAN | OPRD1 | P41143 | CHEMBL236 | 10731 / 12871 |
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 | opioid receptor kappa 1 | Homo sapiens; Human | OPRK_HUMAN | OPRK1 | P41145 | CHEMBL237 | 11463 / 13975 |
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 | opioid receptor mu 1 | Homo sapiens; Human | OPRM_HUMAN | OPRM1 | P35372 | CHEMBL233 | 12998 / 15406 |
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 | opioid related nociceptin receptor 1 | Homo sapiens; Human | OPRX_HUMAN | OPRL1 | P41146 | CHEMBL2014 | 3236 / 3473 |
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 | platelet activating factor receptor | Homo sapiens; Human | PTAFR_HUMAN | PTAFR | P25105 | CHEMBL250 | 822 / 2569 |
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 | trace amine associated receptor 1 | Homo sapiens; Human | TAAR1_HUMAN | TAAR1 | Q96RJ0 | CHEMBL5857 | 1333 / 1340 |
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 | thyroid stimulating hormone receptor | Homo sapiens; Human | TSHR_HUMAN | TSHR | P16473 | CHEMBL1963 | 29918 / 29937 |
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 | arginine vasopressin receptor 1A | Homo sapiens; Human | V1AR_HUMAN | AVPR1A | P37288 | CHEMBL1889 | 2156 / 3971 |
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 | vasoactive intestinal peptide receptor 1 | Homo sapiens; Human | VIPR1_HUMAN | VIPR1 | P32241 | CHEMBL5144 | 148 / 1892 |
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